Day 1

All times shown in CEST

Recordings are passcode-protected (registrants only)

9:00 - 10:30

Welcome & Opening

Virtual Get Together

Chairs: Jana Selent & Miriam Scarpa

Session 1: Keynote Lecture 1

Chair: Andreas Bock

Arun Shukla (Indian Institute of Technology, Kanpur, Uttar Pradesh, India)

Intrinsic bias at non-canonical, β-arrestin-coupled seven transmembrane receptors

(not recorded upon request)

15 min Break

Join us for Networking!

10:45 - 12:00

Session 2: Signaling Map

An overview on signaling map activities

Chairs: Marcel Bermúdez & Jana Selent

Avgi Apostolakou (University of Athens, Greece)

The extended human GPCR network: hGPCRnet

Irene Coin (University of Leipzig, Germany)

Live-cell structural insights into arrestin interactions with a secretin-like GPCR

Tõnis Laasfeld (University of Tartu, Estonia)

Imaging artifacts and how to find them? Impact of artifacts on quantitative microscopy-based GPCR measurements

Abigail Pearce (University of Cambridge, UK)

Negative regulation of Calcitonin-Like Receptor signalling by β-arrestin and GRK expression

Flash Poster Talks 1

Pre-recorded 3 minute talks selected from submitted abstracts

Chairs: Miriam Scarpa & Jose Andres Alepuz Guillen

1.1 André Dias (University of Copenhagen, Denmark)

Can you further improve the experimental conditions of your cellular assays? - The case of ligand binding

1.2 Kristina Puls (Freie Universität Berlin, Germany)

Enlightenment Through Dynamics: How the Peripheral Analgesic HS-731 Discriminates Between Opioid Receptors

1.3 Amlan Ganguly (Institute of Molecular, Cell and Systems Biology, University of Glasgow, UK)

The role of disulphide bonds in the extracellular domain of isoforms of human GPR35

1.4 Amandeep Kaur Gill (Queen Mary University of London, UK)

​Probe Confined Dynamic Mapping for GPCR Allosteric Site Prediction

1.5 Maria Majellaro (Celtarys Research, & University of Santiago de Compostela, Spain)

Novel fluorescent probes for the characterization of Cannabinoid Receptors through diverse fluorescence-based assays

1.6 Sébastien Fiorucci (Université Côte d’azur, France)

Structure-based virtual screening of bitter taste receptors

1.7 Carole Daly (Queen’s University Belfast, UK)

G protein selectivity and gene regulation by US28 are shaped by the presence or absence of chemokines

1.8 Pietro Cocchiara (Institute of Molecular, Cell and Systems Biology, University of Glasgow, UK)

IT1t antagonizes and regulates the oligomerization state of CXCR4

1.9 Lisa Reinmuth (University of Copenhagen, Denmark)

GPR183 receptor-ligand interactions – In silico and in vitro screening of an endogenous ligand and small molecule agonists in development

1.10 Sabina Podlewska (Maj Institute of Pharmacology Polish Academy of Sciences, Poland)

Generation of new potential CYP inhibitors via automated structure modification and docking

12:40 - 14:00

Networking and Lunch

Opportunity to network and visit poster presenters in Wonder

15 min Break

Join us for Networking!

(Session has been cancelled)

Yamina Berchiche (Dr. GPCR)

Dr. GPCR Ecosystem 2.0: Collaborating Better

17:00 - open end